Tsev - Cov khoom - Peptide - Paub meej
Retatrutide Powder CAS .2381089-83-2 98% Purity Min
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Retatrutide Powder CAS .2381089-83-2 98% Purity Min

Retatrutide Powder CAS .2381089-83-2 98% Purity Min

Lub npe Askiv: Retatrutide
CAS Nr .: 2381089-83-2
Molecular Luj: 4813.58g/mol
Molecular Formula: C₂₂₁H₃4₉N₆₅O₇₁S
Qhov tsos: dawb hmoov
tsw: no
Stability: ruaj khov
MSDS thiab COA: muaj rau koj siv
Peev xwm: 500g ib hlis
Qhov tsos: dawb hmoov
Source: hluavtaws
Purity (HPLC) >98.0%
Qhov chaw ntawm Keeb Kwm: Tuam Tshoj Yinherb-Lab
Packing: Raws li tus neeg siv khoom xav tau
Yam tsawg kawg nkaus Order Quantity: 10g
Cia: Khaws rau hauv qhov chaw txias & qhuav, Khaws kom deb ntawm lub teeb muaj zog thiab cua sov rau 2 xyoos

Hauj lwm lawm

Xi'an Yinherb Bio-Tech Co., Ltd. yog ib qho ntawm cov ua lag luam thiab cov chaw muag khoom ntawm rettrutide hmoov cas.2381089-83-2 98% purity min hauv Suav teb, kuj txhawb kev pabcuam customized. Zoo siab txais tos mus yuav bulk retatrutide hmoov cas.2381089-83-2 98% purity min rau muag ntawm no los ntawm peb lub hoobkas. Cov khoom zoo thiab tus nqi tsim nyog muaj.

 

 

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Kev Tshawb Fawb Kev Tshawb Fawb ntawm Nootropics & peptide hauv Suav teb

Yinherb Lab yog lub chaw tshawb fawb kev tshaj lij hauv Suav teb, tau tsom mus rau Cov Khoom Noj Khoom Haus, Nootropics thiab Peptide raw cov ntaub ntawv tshawb fawb thiab tsim tawm hauv kev lag luam no rau ntau tshaj 10 xyoo nrog kev ruaj khov zoo thiab muaj koob npe nrov, peb tuaj yeem muab txhua qhov kev xeem batch, suav nrog COA, HPLC thiab NMR. Kuv ntseeg tias peb yuav tsum ua haujlwm zoo yav tom ntej.

Yinherb Lab High Quality Retatrutide Powder CAS{0}}% Purity Min

Khoom npe:

Retatrutide  
CAS Nr 2381089 - 83 - 2 Pharmacological Assay
Molecular Formula C₂₂₃H₃₄₃F₃N₄₆O₇₀ Edman Degradation / Mass Spectrometry (MS)
Molecular Luj 4845.444 g·mol⁻¹ Elemental Analysis & NMR
Cov yam ntxwv zoo Nws yog 39 - amino - acid hluavtaws peptide tsim los ntawm GIP peptide qaum. Nws muaj peb yam tsis yog - tus qauv amino acids los txhim kho kev ruaj ntseg. Nws muaj kev sib raug zoo rau GIP receptor (8.9 npaug ntau dua qhov muaj zog dua li glucagon thiab GLP - 1 receptors), thiab nws cov qauv molecular tshwj xeeb ua rau nws ua tau zoo rau peb qhov tseem ceeb metabolic receptors. Electrospray Ionization Mass Spectrometry (ESI{0}}MS)
Qhov tshwm sim Dawb kom tawm -dawb, dawb- ntws lyophilized hmoov; tsw tsw Kev soj ntsuam pom pom & Olfactory (USP<191>)
Purity (HPLC) Ntau dua lossis sib npaug li 99.0% (API Qib); Yam Khoom Muaj Tsawg dua lossis sib npaug li 1.0% RP-HPLC (USP<621>, Kem: C18, Mobile Phase: Acetonitrile-Dej-Trifluoroacetic Acid)
Solubility Soluble hauv dej (Ntau dua lossis sib npaug ntawm 20 mg / mL, 25 degree); me ntsis soluble hauv ethanol; insoluble nyob rau hauv non-polar solvents Gravimetric Solubility Test (EP 2.2.10)
Isoelectric Point (pI) 8.5–9.0 Isoelectric Focusing Electrophoresis
Kev ua lom lom EC₅₀ rau GIP Receptor: Tsawg dua lossis sib npaug rau 0.5 nM; EC₅₀ rau GLP-1 Receptor: Tsawg dua lossis sib npaug rau 0.3 nM Cell -Raws li Kev Ntsuas Ua Haujlwm (cAMP Detection)
Poob rau ziab Tsawg dua lossis sib npaug li 2.0% Nqus Qhuav ntawm 60℃rau 3h (USP<731>)
Hnyav Hlau Tag nrho cov hlau hnyav tsawg dua lossis sib npaug li 5 ppm; Lead (Pb) Tsawg dua lossis sib npaug li 1 ppm; Cadmium (Cd) Tsawg dua lossis sib npaug li 0.1 ppm ICP-MS (USP<233>)
Cov ntsiab lus Endotoxin Tsawg dua lossis sib npaug li 0.5 EU / mg Limulus Amebocyte Lysate (LAL) Test (USP<85>)
Microbial txwv Tag nrho Aerobic Microbial suav Tsawg dua lossis sib npaug rau 10 CFU / g; Pwm & Pwm Tsawg dua lossis sib npaug li 5 CFU / g; Cov kab mob (E. coli, Salmonella) Tsis zoo USP<61> & <62>

Retatrutide Powder yog dab tsi?

Retatrutide (code: LY-3437943) yog ib qho kev sim peptide tshuaj tsim los ntawm Eli Lilly, uas sawv cev rau kev uatriple agonist ntawm GLP - 1, GIP, thiab glucagon receptors. Nws qhia tau hais tias muaj txiaj ntsig zoo tshaj plaws hauv kev poob phaus thiab kev tswj ntshav qab zib, thiab tam sim no nyob rau hauv lig - theem kev soj ntsuam, nrog rau qhov dav dav hauv kev kho mob rog rog thiab ntshav qab zib hom 2.

Nws yog feem ntau nthuav tawm raws li cov hmoov dawb. Nws yuav tsum tau muab khaws cia rau ntawm - 20℃lossis qis dua hauv lub xeev lyophilized los tiv thaiv kev degradation thiab tuav nws txoj haujlwm lom neeg.

 

Nws ib nrab - lub neej yog li 6 hnub, thiab lub sijhawm kom ncav cuag cov ntshav siab tshaj plaws yog 8 - 72 teev. Lub bioavailability ntawm kev txhaj tshuaj subcutaneous yog 80%, thiab nws tuaj yeem muab tshuaj ib zaug ib lim tiam.

Oligopeptide - 1 17

product-1-1

 

Retatrutide Powder Mechanism ntawm Kev Ua thiab Kev Ua Haujlwm Ntxiv

Nws ua kom muaj kev sib koom ua ke ntawm kev tswj hwm ntawm cov metabolism los ntawm ib txhij ua kom peb cov tshuaj hormones receptors, uas muaj ntau dua li cov tshuaj ib leeg lossis dual agonist:

GLP - 1 Receptor Activation: Nws tuaj yeem ua rau lub plab zom mov qeeb, txhawb nqa cov piam thaj - nyob ntawm insulin tso tawm, inhibit glucagon tso tawm ntau dhau, thiab txhim kho satiety, yog li txo cov khoom noj.

 

GIP Receptor Activation: Nws ua kom lub cev lub cev cov tshuaj insulin tom qab noj mov, txhim kho cov metabolism hauv lipid, thiab pab ntxiv rau hauv stabilizing ntshav qab zib thiab txo cov rog.

 

Glucagon Receptor Activation: Nws txhawb nqa lub cev lipolysis txheej txheem, hloov cov roj cia rau hauv lub zog, ua kom lub zog noj txhua hnub, thiab ua kom cov rog tsis tau yooj yim ua rau cov leeg nqaij.

 

retatrutide


Retatrutide Powder Application Scenarios thiab Kev Siv Cov Cai

Nws txoj kev ua tau zoo tau raug tshawb xyuas tag nrho hauv Phase 2 kev sim tshuaj ntsuam xyuas kev rog rog thiab hom 2 mob ntshav qab zib:

 

Kev rog rog: Hauv kev sim nrog 338 cov neeg laus rog rog lossis rog rog, tom qab 48 lub lis piam ntawm kev txhaj tshuaj subcutaneous txhua lub limtiam, qhov kev poob phaus yog koob tshuaj - nyob ntawm. Pab pawg koob tshuaj 12mg tau ua tiav qhov hnyav nruab nrab ntawm 24.2%, thiab pawg 8mg koob ua tiav 22.8%. Txhua tus neeg koom nrog hauv pawg siab - koob tshuaj poob ntau dua 5% ntawm lawv qhov hnyav, thiab 75% - 83% poob ntau dua 15% ntawm lawv qhov hnyav. Lub caij no, cov neeg tuaj koom tau txo qis ntawm 600 calories hauv kev noj txhua hnub.

 

Hom 2 Ntshav Qab Zib: Hauv kev sim nrog 281 tus neeg mob ntshav qab zib hom 2, nws tsis tsuas yog txo cov neeg mob qhov hnyav xwb tab sis kuj txo qis HbA1c thiab ceev cov ntshav qabzib. Tsis tas li ntawd, nws kuj tau txhim kho cov kab mob plawv xws li ntshav siab, triglycerides, thiab cov roj cholesterol.

 

Tsis yog - cawv Fatty Liver Disease: Ib txoj kev tshawb fawb 2024 tau qhia tias nws tuaj yeem txo cov rog rog los ntawm 82.4% tom qab 24 lub lis piam ntawm kev siv, uas qhia tau tias nws muaj peev xwm kho cov kab mob metabolic - ntsig txog kab mob siab.

 

Retatrutide Powder Storage Conditions

Ntim Specifications: Lyophilized hmoov ntim rau hauv 1g / vial, 5g / vial, los yog 10g / vial (amber iav vials nrog roj hmab stoppers thiab txhuas crimp seals) los tiv thaiv lub teeb thiab noo noo. Ntim ntim rau kev lag luam siv: 100g / nruas (txhuas-kab HDPE nruas).

 

Kev cia khoom: Khw ntawm-20℃± 5 degreenyob rau hauv ib lub thawv ntim, lub teeb - tiv thaiv; zam rov qab khov -thaw cycles. Txee lub neej: 24 lub hlis raws li kev pom zoo cia (validated ntawm ICH Q1A stability test).

 

Cov khoom muaj feem xyuam

Tshwj xeeb hauv Semaglutide, Tirzepatide, Retatrutide, DSIP, Eptalone, Selank, Semax, Melanotan II, Thymosin alpha 1, Oxytocin, P21, Adamax, Dihexa thiab tus tub ntawm.

  • Myristoyl Tetrapeptide-12

    Yinherb
     
  • Palmitoyl Tripeptide-1

    Yinherb
  • Acetyl Tetrapeptide-2

    Yinherb
  • Hexapeptide-9

    Yinherb
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Cov ntawv pov thawj

 

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FDA

product-650-920

Halal

product-650-927

ISO 9001 Cov

product-650-920

Kosher

product-3969-5613

Kev Tshawb Fawb Tshaj Tawm

product-3969-5613

SGS

 

 

Yinherb Lab nrhiav tau nyob rau hauv 2009, tau mob siab rau rau biotechnology teb rau ntau tshaj kaum xyoo. Niaj hnub no, nws tau tsim ib qho kev txhim kho kev ua haujlwm nrog "R & D + ntau lawm" ua ib qho kev sib koom ua ke. Thiab ib txwm ua raws li cov kev lag luam tseem ceeb ntawm "Quality First, Service Second, Price Third".

Peb qhov chaw nyob

No.3, Daqing rd, Hi-tech zone, Xi'an nroog, Suav teb.

Xov tooj

+8618681897250

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Cim npe nrov: Retatrutide hmoov cas.2381089-83-2 98% purity min, Tuam Tshoj rettrutide hmoov cas.2381089-83-2 98% purity min manufacturers, lwm tus neeg, Hoobkas

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